Centella Asiatica Extract

Botanical Anti-inflammatory

Also known as: Cica, Gotu Kola, Madecassoside, Asiaticoside

Description

Centella asiatica is a herbaceous plant used for centuries in Ayurvedic and traditional medicine. Its dermatological activity is attributed to four key triterpenoid saponins: madecassoside, asiaticoside, asiatic acid, and madecassic acid (collectively known as centelloids). These compounds stimulate type I and III collagen synthesis, promote fibroblast proliferation, inhibit inflammatory cytokines, and accelerate wound healing. Centella extract is widely used in Korean skincare ('Cica' products) for calming sensitive, irritated, and acne-prone skin.

Mechanism of Action

Asiaticoside and madecassoside stimulate collagen synthesis by activating the TGF-β/Smad signaling pathway in dermal fibroblasts and upregulating type I procollagen gene expression. Asiatic acid increases antioxidant enzyme activity (SOD, catalase, glutathione peroxidase) and inhibits NF-κB-mediated pro-inflammatory cytokine production (TNF-α, IL-1β, IL-6). Madecassoside promotes angiogenesis and re-epithelialization in wound models. Together, centelloids modulate both the inflammatory and proliferative phases of tissue repair.

Indications

  • Wound healing and scar management
  • Acne and post-acne erythema
  • Sensitive or irritated skin
  • Rosacea-prone skin
  • Photoaging / fine lines
  • Atopic dermatitis adjunct
  • Post-procedural recovery
  • Stretch marks (striae)

Available Concentrations

0.1% (titrated extract — TECA)1%2%5%10%

Side Effects

  • Allergic contact dermatitis (uncommon; sensitization to triterpenoid fraction)
  • Mild irritation in rare cases

Contraindications

  • Known hypersensitivity to Centella asiatica or its triterpenoids
  • History of allergic contact dermatitis to Centella-containing products

Pregnancy Category

Not classified (insufficient data; generally considered safe for topical use at cosmetic concentrations)

Found In

Cosmetics containing Centella Asiatica Extract

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